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Examples
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The interesting thing is that when you study the distribution based on RNase, you find that all the active-site residues were conserved after gene duplication, as was the RNA-binding site.
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As per protocol, dose escalation will continue up to three levels above full Btk active-site occupancy, which occurred in dose cohort 2.
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Correlating kinase active-site occupancy with efficacy.
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Correlating kinase active-site occupancy with efficacy.
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Correlating kinase active-site occupancy with efficacy.
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With the classical, active-site oriented drug-development approach reaching its limits, protein ligand-binding sites in general and allosteric sites in particular are increasingly attracting the interest of medicinal chemists in the search for new types of targets and strategies to drug development.
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As per protocol, dose escalation will continue up to three levels above full Btk active-site occupancy, which occurred in dose cohort 2.
THE MEDICAL NEWS Editors 2010
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With the classical, active-site oriented drug-development approach reaching its limits, protein ligand-binding sites in general and allosteric sites in particular are increasingly attracting the interest of medicinal chemists in the search for new types of targets and strategies to drug development.
BioMed Central - Latest articles Alejandro Panjkovich 2010
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Through protein-protein interactions, the regulatory protein can remodel the active-site cavity of the catalytic protein for synthesizing the precursor of menthol, which is released from the plant as mint scent.
Taipei Times 2010
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With the classical, active-site oriented drug-development approach reaching its limits, protein ligand-binding sites in general and allosteric sites in particular are increasingly attracting the interest of medicinal chemists in the search for new types of targets and strategies to drug development.
BioMed Central - Latest articles Alejandro Panjkovich 2010
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